CAS Number 342882-77-3 IUPHAR/BPS 732 Formula C26H42N2O2 Molar mass 414.622 g/mol | PubChem CID 9823107 ChemSpider 7998855 3D model (Jmol) Interactive image | |
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O-1812 is an eicosanoid derivative related to anandamide that acts as a potent and highly selective agonist for the cannabinoid receptor CB1, with a Ki of 3.4 nM at CB1 and 3870 nM at CB2. Unlike most related compounds, O-1812 is metabolically stable against rapid breakdown by enzymes, and produces a cannabinoid-like discriminative effect in rats, which is similar but not identical to that produced by cannabinoid drugs of other chemical classes.
References
O-1812 Wikipedia(Text) CC BY-SA