ATC code None PubChem CID 5387 Formula C19H22N4O2S Molar mass 370.47 g/mol ChEMBL ID 253978 | CAS Number 80880-90-6 UNII 0990EG3K10 3D model (Jmol) Interactive image Pubchem 5387 ChemSpider ID 5194 | |
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M2 receptors labelled with cy3b telenzepine myocytes in mouse heart slice 23oc
Telenzepine is a thienobenzodiazepine acting as selective M1 antimuscarinic. It is used in the treatment of peptic ulcers. Telenzepine is atropisomeric, in other words the molecule has a stereogenic C–N-axis; in neutral aqueous solution it displays a half-life for racemization of the order of 1000 years. The enantiomers have been resolved. The activity is related to the (+)-isomer which is about 500-fold more active as the (–)-isomer at muscarinic receptors in the rat cerebal cortex.
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How to pronounce telenzepine
References
Telenzepine Wikipedia(Text) CC BY-SA