Harman Patil (Editor)

SRX246

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ATC code
  
None

Formula
  
C42H49N5O5

Molar mass
  
703.88 g/mol

CAS Number
  
512784-93-9

3D model (Jmol)
  
Interactive image

SRX246 httpsuploadwikimediaorgwikipediacommonsthu

SRX246, also known as API-246, is a small-molecule, centrally-active, highly-selective vasopressin V1A receptor antagonist which is under investigation by Azevan Pharmaceuticals for the treatment of affective and anger disorders. It is an azetidinone derivative, and was developed from LY-307174 as a lead compound. A phase II activity trial of the drug in the treatment of adults with intermittent explosive disorder is ongoing. It is also being studied for the treatment of post-traumatic stress disorder.

References

SRX246 Wikipedia