Trisha Shetty (Editor)

Raseglurant

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ATC code
  
None

PubChem CID
  
10331863

Formula
  
C15H13FN2

Molar mass
  
240.276 g/mol

CAS Number
  
757950-09-7

ChemSpider
  
8507323

3D model (Jmol)
  
Interactive image

Raseglurant httpsuploadwikimediaorgwikipediacommonsthu

Raseglurant (INN) (code name ADX-10059) is a negative allosteric modulator of the mGlu5 receptor and derivative of MPEP which was under development by Addex Therapeutics for the treatment of migraine, gastroesophageal reflux disease, and dental anxiety. It reached phase II clinical trials for all of the aforementioned indications before being discontinued due to the observation of possible predictive signs of hepatotoxicity in patients with long-term use.

References

Raseglurant Wikipedia