Synonyms PEAQX, NVP-AAM077 Formula C17H17BrN3O5P Molar mass 454.211 g/mol ChemSpider ID 8044242 | PubChem CID 9868551 3D model (Jmol) Interactive image Pubchem 9868551 | |
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PEAQX is a competitive antagonist at the NMDA receptor. Although originally described as 100-fold selective for GluN1/GluN2A receptors vs. GluN1/GluN2B receptors, more detailed studies of the Ki of PEAQX revealed it only shows a 5 fold difference in affinity for GluN1/GluN2A vs. GluN1/GluN2B receptors. It is also a potent anticonvulsant in animal tests.
References
PEAQX Wikipedia(Text) CC BY-SA