CAS Number 138356-12-4 ChemSpider 7972689 3D model (Jmol) Interactive image | PubChem CID 9796923 Formula C16H24Cl2N2 Molar mass 315.28 g/mol | |
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BD1067 or N-[2-(3,4-dichlorophenyl)ethyl]-N-ethyl-1-pyrrolidineethanamine is a selective sigma receptor antagonist, with a reported binding affinity of Ki = 2 ± 0.5 nM for the sigma-1 receptor and greater than 19 times selectivity over the sigma-2 receptor.
Like other sigma receptor antagonists, pretreating Swiss Webster mice with BD1067 significantly attenuates the behavioral toxicity of cocaine.
References
BD1067 Wikipedia(Text) CC BY-SA