Neha Patil (Editor)

BD1052

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CAS Number
  
138356-16-8

ChemSpider
  
7973202

3D model (Jmol)
  
Interactive image

PubChem CID
  
9797436

Formula
  
C17H24Cl2N2

Molar mass
  
327.294 g/mol

BD1052

BD1052 or N-[2-(3,4-dichlorophenyl)ethyl]-N-2-propen-1-yl-1-pyrrolidineethanamine is a selective sigma receptor agonist, with a reported binding affinity of Ki = 2 ± 0.5 nM for the sigma-1 receptor and 30 times selectivity over the sigma-2 receptor.

Consistent with other reported sigma receptor agonists, pretreating Swiss Webster mice with BD1052 significantly increases the behavioral toxicity of cocaine.

References

BD1052 Wikipedia