Puneet Varma (Editor)

5 HT1F receptor

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Species
  
Human

Entrez
  
3355

Human
  
Mouse

Ensembl
  
ENSG00000179097

5-HT1F receptor

Aliases
  
HTR1F, 5-HT-1F, 5-HT1F, 5HT6, HTR1EL, MR77, 5-HT1F receptor, 5-hydroxytryptamine receptor 1F

External IDs
  
MGI: 99842 HomoloGene: 37361 GeneCards: HTR1F

5-hydroxytryptamine (serotonin) receptor 1F, also known as HTR1F is a 5-HT1 receptor protein and also denotes the human gene encoding it.

Contents

Agonists

  • 5-n-Butyryloxy-DMT: >60-fold selectivity versus 5-HT1E receptor
  • BRL-54443 - mixed 5-HT1E/1F agonist
  • Eletriptan - mixed 5-HT1B/1D/1E/1F/2B/7 agonist
  • LY-334,370 - as well as related benzamides
  • LY-344,864 (N-[(3R)-3-(Dimethylamino)-2,3,4,9-tetrahydro-1H-carbazol-6-yl]-4-fluorobenzamide)
  • Naratriptan - mixed 5-HT1B/1D/1F agonist
  • Antagonists

    MLS000756415

    References

    5-HT1F receptor Wikipedia