Samiksha Jaiswal (Editor)

Zenazocine

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ATC code
  
None

PubChem CID
  
9885108

3D model (Jmol)
  
Interactive image

Pubchem
  
9885108

CAS Number
  
74559-85-6

Formula
  
C23H35NO2

Molar mass
  
357.53 g/mol

ChemSpider ID
  
8060782

Zenazocine httpsuploadwikimediaorgwikipediacommonsthu

Legal status
  
In general: non-regulated

Zenazocine (INN; WIN-42,964) is an opioid analgesic of the benzomorphan family which made it to phase II clinical trials before development was ultimately halted and it was never marketed. It acts as a partial agonist of the μ- and δ-opioid receptors, with less intrinsic activity at the former receptor and more at the latter receptor (hence, it behaves more antagonistically at the former and more agonistically at the latter), and produces antinociceptive effects in animal studies.

References

Zenazocine Wikipedia