PubChem CID 42633508 Molar mass 351.276 g/mol ChEMBL ID 466253 | Formula C17H12F3NO4 Pubchem 42633508 ChemSpider ID 24606034 | |
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VU-0238429 is a drug which acts as a selective positive allosteric modulator for the muscarinic acetylcholine receptor M5. It was the first selective ligand developed for the M5 subtype, and is structurally derived from older M1-selective positive allosteric modulators such as VU-0119498. Replacing the O-methyl- by a phenylgroup further improves the receptor subtype selectivity (VU-0400265).
References
VU-0238429 Wikipedia(Text) CC BY-SA