Kalpana Kalpana (Editor)

Tanaproget

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ATC code
  
none

CAS Number
  
304853-42-7

DrugBank
  
DB04787

Molar mass
  
297.375 g/mol

Legal status
  
Investigational

PubChem CID
  
4369524

ChemSpider
  
3572060

Tanaproget httpsuploadwikimediaorgwikipediacommonsthu

Tanaproget (INN; developmental code names NSP-989, WAY-166989) is an investigational non-steroidal progestin. It is a high affinity, high efficacy, and very selective agonist of the progesterone receptor (PR). Due to its much more selective binding profile relative to most conventional, steroidal progestins, tanaproget may prove to produce fewer side effects in comparison. As of December 2010, it is in phase II clinical trials in the process of being developed for clinical use as a contraceptive by Ligand Pharmaceuticals.

An analog of tanaproget, 4-fluoropropyltanaproget (18F), has been developed as a radiotracer for imaging of the PR in positron emission tomography.

References

Tanaproget Wikipedia


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