Supriya Ghosh (Editor)

TC OT 39

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ATC code
  
none

3D model (Jmol)
  
Interactive image

Molar mass
  
600.78 g/mol

CAS Number
  
479232-57-0

Formula
  
C32H40N8O2S

ChemSpider ID
  
23249746

TC OT 39 httpsuploadwikimediaorgwikipediacommonsthu

IUPAC ID
  
(2S)-N-[[4-[(4,10-dihydro-1-methylpyrazolo[3,4-b][1,5]benzodiazepin-5(1H)-yl)carbonyl]-2-methylphenyl]methyl]-2-[(hexahydro-4-methyl-1H-1,4-diazepin-1-yl)thioxomethyl]-1-pyrrolidinecarboxamide

TC OT 39 is a non-peptide partial agonist of the oxytocin and vasopressin V2 receptors (Ki = 147 nM and >1000 nM, respectively) and antagonist of the vasopressin V1A receptor (Ki = 330 nM).

References

TC OT 39 Wikipedia
(Text) CC BY-SA