Synonyms RS-127,445 PubChem CID 196968 ChemSpider 170590 Molar mass 281.327 g/mol | CAS Number 199864-87-4 IUPHAR/BPS 188 UNII 0JAU3P8OBM | |
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RS-127445 is a drug which acts as a potent and selective antagonist at the serotonin 5-HT2B receptor, with around 1000x selectivity over the closely related 5-HT2A and 5-HT2C receptors. The role of the 5-HT2B receptor in the body is still poorly understood, and RS-127445 has been a useful tool in unravelling the function of the various systems in which this receptor is expressed.
References
RS-127445 Wikipedia(Text) CC BY-SA