Kalpana Kalpana (Editor)

Perzinfotel

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ATC code
  
none

PubChem CID
  
6918236

UNII
  
FX5AUU7Z8T

Molar mass
  
260.184 g/mol

CAS Number
  
144912-63-0

ChemSpider
  
5293443

KEGG
  
D05447

Perzinfotel httpsuploadwikimediaorgwikipediacommonsthu

Perzinfotel (EAA-090) is a drug which acts as a potent NMDA antagonist. It has neuroprotective effects and has been investigated for the treatment of stroke, but lacks analgesic effects. Nevertheless, it shows a good safety profile compared to older drugs, although further development of this drug has been discontinued.

Prodrugs were developed since the oral bioavailability of perzinfotel is only around 3-5%.

References

Perzinfotel Wikipedia