Puneet Varma (Editor)

PF 514273

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CAS Number
  
851728-60-4

ChemSpider
  
9491886

3D model (Jmol)
  
Interactive image

PubChem CID
  
11316919

Formula
  
C21H17Cl2F2N3O2

Molar mass
  
452.281 g/mol

PF-514273 httpsuploadwikimediaorgwikipediacommonsthu

PF-514273 is a drug developed by Pfizer, which acts as an extremely selective antagonist for the CB1 receptor, with approximately 10,000x selectivity over the closely related CB2 receptor. This very high selectivity makes it useful for scientific research into these receptors, as many commonly used cannabinoid receptor antagonists also block the CB2 receptor to some extent.

References

PF-514273 Wikipedia