Puneet Varma (Editor)

ICI 199,441

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CAS Number
  
115199-84-3

ChemSpider
  
2340095

Formula
  
C21H24Cl2N2O

Molar mass
  
391.333 g/mol

PubChem CID
  
3082718

ChEMBL
  
CHEMBL38576

3D model (Jmol)
  
Interactive image

ICI-199,441 httpsuploadwikimediaorgwikipediacommonsthu

ICI-199,441 is a drug which acts as a potent and selective κ-opioid agonist, and has analgesic effects. It is a biased agonist of the KOR, and is one of a relatively few KOR ligands that is G protein-biased rather than β-arrestin-biased.[1]

References

ICI-199,441 Wikipedia