Puneet Varma (Editor)

GR 127935

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ATC code
  
none

PubChem CID
  
107780

ChEMBL
  
CHEMBL15928

Molar mass
  
497.587 g/mol

CAS Number
  
148672-13-3

IUPHAR/BPS
  
14

Formula
  
C29H31N5O3

GR-127935 httpsuploadwikimediaorgwikipediacommonsthu

GR-127935 is a drug which acts as a selective antagonist at the serotonin receptors 5-HT1B and 5-HT1D. It has little effect when given by itself but blocks the antiaggressive effect of 5-HT1B agonists, and alters release of serotonin in the brain, as well as reducing drug-seeking behaviour in cocaine addicted rats.

References

GR-127935 Wikipedia