CAS Number 144625-51-4 IUPHAR/BPS 247 Formula C19H27N3O4S Molar mass 393.499 g/mol | PubChem CID 119376 ChemSpider 106623 3D model (Jmol) Interactive image | |
![]() | ||
GR-113808 is a drug which acts as a potent and selective 5-HT4 serotonin receptor antagonist. It is used in researching the roles of 5-HT4 receptors in various processes, and has been used to test some of the proposed therapeutic effects of selective 5-HT4 agonists, such as for instance blocking the nootropic effects of 5-HT4 agonists, and worsening the respiratory depression produced by opioid analgesic drugs, which appears to be partly 5-HT4 mediated and can be counteracted by certain 5-HT4 agonists.
References
GR-113808 Wikipedia(Text) CC BY-SA