Harman Patil (Editor)

Casopitant

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ATC code
  
A04AD13 (WHO)

PubChem CID
  
23725089

UNII
  
3B03KPM27L

CAS Number
  
414910-27-3

ChemSpider
  
25069049

Molar mass
  
616.26 g/mol

Casopitant httpsuploadwikimediaorgwikipediacommonsthu

Synonyms
  
(2R,4S)-4-(4-Acetylpiperazin-1-yl)-N-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethyl}-2-(4-fluoro-2-methylphenyl)-N-methylpiperidine-1-carboxamide

How to pronounce casopitant


Casopitant (INN, tentative trade names Rezonic (U.S.), Zunrisa (Europe)) is an neurokinin 1 receptor (NK1R) antagonist undergoing research for the treatment of chemotherapy-induced nausea and vomiting (CINV). It is currently under development by GlaxoSmithKline (GSK).

In July 2008, the company filed a marketing authorisation application with the European Medicines Agency. The application was withdrawn in September 2009 because GSK decided that further safety assessment was necessary.

References

Casopitant Wikipedia