Neha Patil (Editor)

AM 2233

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CAS Number
  
444912-75-8

ChemSpider
  
8401830

ECHA InfoCard
  
100.233.382

PubChem CID
  
10226340

ChEMBL
  
CHEMBL364266

Molar mass
  
458.334 g/mol

AM-2233 httpsuploadwikimediaorgwikipediacommonsthu

Legal status
  
CA: Schedule IIDE: Anlage II (Prohibited)NZ: Temporary Class

AM-2233 is a drug that acts as a highly potent full agonist for the cannabinoid receptors, with a Ki of 1.8 nM at CB1 and 2.2 nM at CB2 as the active (R) enantiomer. It was developed as a selective radioligand for the cannabinoid receptors and has been used as its 131I derivative for mapping the distribution of the CB1 receptor in the brain. AM-2233 was found to fully substitute for THC in rats, with a potency lower than that of JWH-018 but higher than WIN 55,212-2.

As of October 2015 AM-2233 is a controlled substance in China.

References

AM-2233 Wikipedia
(Text) CC BY-SA


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